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Research Interests
Efficient intracellular electron transfer is essential to organisms
that use oxygen. An exquisite balance between oxidized and reduced
enzymes and cofactors, termed redox homeostasis, must be carefully
regulated to maintain cellular function. Loss of redox balance underlies
molecular changes associated with aging and age related diseases.
Consequences of acute or chronic disruption in redox homeostasis
include neurodegenerative diseases, cancer, diabetes mellitus, atherosclerosis,
and rheumatoid arthritis.
In our lab, we are studying the enzymes that control
the levels of thioredoxin
(Trx) and glutathione
(GSH), the major thiol based redox buffer systems.
These parallel yet distinct systems are essential in cellular processes
such as detoxification of reactive oxygen and nitrogen species,
nucleotide biosynthesis, modulation of protein function, and cellular
signaling of apoptosis and differentiation. Despite intensive research
in these areas, critical molecular details are lacking that would
facilitate the design of more effective treatments capable of modulating
the intracellular redox state.

In collaboration with Dr.
Melanie Simpson, we are also studying enzymes
involved in hyaluronan production. Hyaluronan, a polymer comprised
of a repeating disaccharide, has been shown to be important in prostate
cancer progression, wound healing, normal heart development and
other critical developmental processes. However, relatively limited
structural and mechanistic information is available for the enzymes
responsible for its biosynthesis and degradation. Specifically,
we are working on
UDP-glucose dehydrogenase (UGDH), which provides
an essential precursor for hyaluronan production, and hyaluronidase
(Hyal), which processes hyaluronan into smaller
pieces with specific biological functions.
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